Reaction Details Report a problem with these data
Target
Genome polyprotein [1973-2419,R2002H]
Ligand
BDBM243449
Substrate
n/a
Meas. Tech.
Transient Transfection Assay
EC50
0.027±n/a nM
Citation
Vandyck, K; Last, SJ; Houpis, IN; Raboisson, PJ Benzimidazole-imidazole derivatives US Patent US9433609 Publication Date 9/6/2016
More Info.:
Target
Name:
Genome polyprotein [1973-2419,R2002H]
Synonyms:
Non-structural protein 5A (NS5A)(R30H) | POLG_HCVCO | Serine protease NS5A (R30H)
Type:
Enzyme
Mol. Mass.:
48686.12
Organism:
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
Description:
aa 1973-2419
Residue:
447
Sequence:
SGSWLRDVWDWICTVLTDFKTWLQSKLLPHLPGVPFFSCQRGYKGVWRGDGIMQTTCPCGAQITGHVKNGSMRIVGPRTCSNTWHGTFPINAYTTGPCTPSPAPNYSRALWRVAAEEYVEVTRVGDFHYVTGMTTDNVKCPCQVPAPEFFTEVDGVRLHRYAPACKPLLREEVTFLVGLNQYLVGSQLPCEPEPDVAVLTSMLTDPSHITAETAKRRLARGSPPSLASSSASQLSAPSLKATCTTRHDSPDADLIEANLLWRQEMGGNITRVESENKVVILDSFEPLQAEEDEREVSVPAEILRRSRKFPRAMPIWARPDYNPPLLESWKDPDYVPPVVHGCPLPPAKAPPIPPPRRKRTVVLSESTVSSALAELATKTFGSSESSAVDSGTATASPDQPSDDGDAGSDVESYSSMPPLEGEPGDPDLSDGSWSTVSEEASEDVVCC