Reaction Details Report a problem with these data
Target
E3 ubiquitin-protein ligase Mdm2 [23-127]
Ligand
BDBM432007
Substrate
n/a
Meas. Tech.
MDM2-p53 Inhibition AlphaScreen
IC50
17.0±n/a nM
Citation
Weinstabl, H; Gollner, A; Ramharter, J; Wunberg, T Spiro[3H-indole-3,2′-pyrrolidin]-2(1H)-one compounds and derivatives as MDM2-P53 inhibitors US Patent US10576064 Publication Date 3/3/2020
More Info.:
Target
Name:
E3 ubiquitin-protein ligase Mdm2 [23-127]
Synonyms:
MDM2 | MDM2-MDMX (aa 23-127) | MDM2_HUMAN
Type:
Oncoprotein
Mol. Mass.:
12198.94
Organism:
Homo sapiens (Human)
Description:
Q00987[23-127]
Residue:
105
Sequence:
EQETLVRPKPLLLKLLKSVGAQKDTYTMKEVLFYLGQYIMTKRLYDEKQQHIVYCSNDLLGDLFGVPSFSVKEHRKIYTMIYRNLVVVNQQESSDSGTSVSENRC