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Target
Tumor protein p53-inducible nuclear protein 2
Ligand
BDBM449138
Substrate
n/a
Meas. Tech.
Radioligand Binding Assay
EC50
180±n/a nM
Citation
 Shoichet, BK; Lin, H; Gmeiner, P; Manglik, A; Kobilka, B; Roth, BL; Dengler, DG MU opioid receptor modulators US Patent  US10702498 Publication Date 7/7/2020 
Target
Name:
Tumor protein p53-inducible nuclear protein 2
Synonyms:
C20orf110 | DOR | Diabetes and obesity-regulated gene | PIG-U | PINH | T53I2_HUMAN | TP53INP2 | p53-inducible protein U
Type:
Protein
Mol. Mass.:
23980.20
Organism:
Human
Description:
Q8IXH6
Residue:
220
Sequence:
MFQRLSSLFFSTPSPPEDPDCPRAFVSEEDEVDGWLIIDLPDSYAAPPSPGAAPAPAGRPPPAPSLMDESWFVTPPACFTAEGPGLGPARLQSSPLEDLLIEHPSMSVYVTGSTIVLEPGSPSPLPDAALPDGDLSEGELTPARREPRAARHAAPLPARAALLEKAGQVRRLQRARQRAERHALSAKAVQRQNRARESRPRRSKNQSSFIYQPCQRQFNY
  
Inhibitor
Name:
BDBM449138
Synonyms:
US10702498, Compound 12 | US11484525, Compound 12
Type:
Small organic molecule
Emp. Form.:
C19H28N3OS
Mol. Mass.:
346.51
SMILES:
C[C@H](Cc1ccsc1)NC(=O)NC[C@@H](Cc1ccccc1)[NH+](C)C |r|
Structure:
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