| Assay Method Information | |
| | ChEMBL_1824965 (CHEMBL4324729) |
| Description: | Non-competitive insurmountable antagonist activity at human CCR5 expressed in human U2OS cell membranes assessed as pEC50 for CCL3-stimulated [35S]GTPgammaS binding at 300 nM preincubated for 30 mins followed by [35S]GTPgammaS addition and measured after 90 mins (Rvb = 8.42 +/- 0.06 No_unit) |
| Affinity data for this assay | |
|---|---|
| If you find an error in this entry please send us an E-mail | |