Assay Method Information

Assay Name:  ChEMBL_1566072 (CHEMBL3791459)
Description:  Competitive inhibition of human KDM4A (1 to 359 residues) expressed in competent Escherichia coli BL21-CodonPlus-RIL cells using 2-oxoglutarate as substrate preincubated for 10 mins followed by substrate addition measured after 45 mins by TR-FRET assay
Affinity data for this assay
 

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