Assay Method Information

Assay Name:  ChEMBL_1824952 (CHEMBL4324716)
Description:  Non-competitive insurmountable antagonist activity at human CCR2 expressed in human U2OS cell membranes assessed as EC50 for CCL2-stimulated [35S]GTPgammaS binding at 10 nM preincubated for 30 mins followed by [35S]GTPgammaS addition and measured after 90 mins (Rvb = 8 nM)
Affinity data for this assay
 

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