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Report error Found 9 Enz. Inhib. hit(s) for PDB: 1OWE
LigandPNGBDBM50138670(6-Carbamimidoyl-naphthalene-2-carboxylic acid phen...)
Affinity DataKi:  628nMAssay Description:Photometric_Method1More data for this Ligand-Target Pair
In DepthDetails D3R
PDB3D3D Structure (crystal)
LigandPNGBDBM50138670(6-Carbamimidoyl-naphthalene-2-carboxylic acid phen...)
Affinity DataKi:  628nM ΔG°:  -35.4kJ/molepH: 7.4 T: 25°CAssay Description:Abbott uPA__Urokinase Human - Ki(uM)More data for this Ligand-Target Pair
LigandPNGBDBM50138670(6-Carbamimidoyl-naphthalene-2-carboxylic acid phen...)
Affinity DataKi:  630nMAssay Description:Binding affinity towards Urokinase-type plasminogen activator (urokinase)More data for this Ligand-Target Pair
LigandPNGBDBM50138670(6-Carbamimidoyl-naphthalene-2-carboxylic acid phen...)
Affinity DataKi:  631nMAssay Description:Inhibition of urokinaseMore data for this Ligand-Target Pair
LigandPNGBDBM50138670(6-Carbamimidoyl-naphthalene-2-carboxylic acid phen...)
Affinity DataKi:  631nMAssay Description:Binding affinity to human urokinase-type plasminogen activator (microPa).More data for this Ligand-Target Pair
LigandPNGBDBM50138670(6-Carbamimidoyl-naphthalene-2-carboxylic acid phen...)
Affinity DataKi:  631nMAssay Description:Binding affinity value against urokinase plasminogen activatorMore data for this Ligand-Target Pair
LigandPNGBDBM50138670(6-Carbamimidoyl-naphthalene-2-carboxylic acid phen...)
Affinity DataKi:  631nMAssay Description:Inhibition of human uPA using pyroGlu-Gly-Arg-p-NA.HCl as substrate preincubated for 15 mins prior sustrate addition measured for 10 mins by spectrop...More data for this Ligand-Target Pair
LigandPNGBDBM50138670(6-Carbamimidoyl-naphthalene-2-carboxylic acid phen...)
Affinity DataKi:  1.90E+3nMAssay Description:Competitive inhibition of human uPA using pyroGlu-Gly-Arg-p-NA.HCl as substrate preincubated for 15 mins prior sustrate addition measured for 10 mins...More data for this Ligand-Target Pair
LigandPNGBDBM50138670(6-Carbamimidoyl-naphthalene-2-carboxylic acid phen...)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of human uPA using pyroGlu-Gly-Arg-p-NA.HCl as substrate preincubated for 15 mins prior sustrate addition measured for 10 mins by spectrop...More data for this Ligand-Target Pair