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11 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Discovery of pyrido[3,4-g]quinazoline derivatives as CMGC family protein kinase inhibitors: Design, synthesis, inhibitory potency and X-ray co-crystal structure.EBI
University of Clermont Auvergne
Perspectives on the Two-Pore Domain Potassium Channel TREK-1 (TWIK-Related K(+) Channel 1). A Novel Therapeutic Target?EBI
University of Clermont Auvergne
Synthesis and biological activity of pyrazole analogues of the staurosporine aglycon K252c.EBI
University of Clermont Auvergne
Synthesis and activities of new indolopyrrolobenzodiazepine derivatives toward acute myeloid leukemia cells.EBI
University of Clermont Auvergne
Synthesis and biological evaluation of Haspin inhibitors: Kinase inhibitory potency and cellular activity.EBI
University of Clermont Auvergne
Synthesis of new pyrazolo[4,3-a]phenanthridine Pim-1 inhibitors and evaluation of their cytotoxic activity towards the MOLM-13 acute myeloid leukemia cell line.EBI
University of Clermont Auvergne
Improved potency of pyridin-2(1H)one derivatives for the treatment of mechanical allodynia.EBI
University of Clermont Auvergne
Pyridin-2(1H)one derivatives: A possible new class of therapeutics for mechanical allodynia.EBI
University of Clermont Auvergne
New pyrido[3,4-g]quinazoline derivatives as CLK1 and DYRK1A inhibitors: synthesis, biological evaluation and binding mode analysis.EBI
University of Clermont Auvergne
Kinase inhibitions in pyrido[4,3-h] and [3,4-g]quinazolines: Synthesis, SAR and molecular modeling studies.EBI
University of Clermont Auvergne
Structure-activity relationship study of hypoxia-activated prodrugs for proteoglycan-targeted chemotherapy in chondrosarcoma.EBI
University of Clermont Auvergne