11 articles for thisTarget
The following articles (labelled with PubMed ID or TBD) are for your review
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Discovery of pyrido[3,4-g]quinazoline derivatives as CMGC family protein kinase inhibitors: Design, synthesis, inhibitory potency and X-ray co-crystal structure.

University of Clermont Auvergne
Perspectives on the Two-Pore Domain Potassium Channel TREK-1 (TWIK-Related K(+) Channel 1). A Novel Therapeutic Target?

University of Clermont Auvergne
Synthesis and biological activity of pyrazole analogues of the staurosporine aglycon K252c.

University of Clermont Auvergne
Synthesis and activities of new indolopyrrolobenzodiazepine derivatives toward acute myeloid leukemia cells.

University of Clermont Auvergne
Synthesis and biological evaluation of Haspin inhibitors: Kinase inhibitory potency and cellular activity.

University of Clermont Auvergne
Synthesis of new pyrazolo[4,3-a]phenanthridine Pim-1 inhibitors and evaluation of their cytotoxic activity towards the MOLM-13 acute myeloid leukemia cell line.

University of Clermont Auvergne
Improved potency of pyridin-2(1H)one derivatives for the treatment of mechanical allodynia.

University of Clermont Auvergne
Pyridin-2(1H)one derivatives: A possible new class of therapeutics for mechanical allodynia.

University of Clermont Auvergne
New pyrido[3,4-g]quinazoline derivatives as CLK1 and DYRK1A inhibitors: synthesis, biological evaluation and binding mode analysis.

University of Clermont Auvergne
Kinase inhibitions in pyrido[4,3-h] and [3,4-g]quinazolines: Synthesis, SAR and molecular modeling studies.

University of Clermont Auvergne
Structure-activity relationship study of hypoxia-activated prodrugs for proteoglycan-targeted chemotherapy in chondrosarcoma.

University of Clermont Auvergne