BDBM152260 US8993552, 1F4 Compound 44

SMILES Cc1nn(nc1C(N)=O)-c1ccccc1

InChI Key InChIKey=IHPOVUXVIZRYAC-UHFFFAOYSA-N

Data  1 IC50  9 Kd

PDB links: 1 PDB ID matches this monomer.

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 152260   

TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM152260(US8993552, 1F4 Compound 44)
Affinity DataKd:  2.50E+5nMAssay Description:Displacement of biotinylated small molecule ligand from His/FLAG-tagged PCAF bromodomain (719 to 832 residues) (unknown origin) after 15 mins by Alph...More data for this Ligand-Target Pair