BDBM179887 US10287250, Compound C.5::US10752592, Compound TABLE C.-9::US9133125, Table C, Compound 5::US9656961, Example 00152
SMILES COCCN1CC[C@]2(C)[C@@H](C)[C@H]1Cc1ccc(O)cc21
InChI Key InChIKey=DZDGGJQZRLCVQI-JCURWCKSSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 179887
Affinity DataKi: 0.110nM ΔG°: -13.6kcal/mole IC50: 26nMpH: 7.5 T: 25°CAssay Description:The Ki (binding affinity) for u opioid receptors was determined using a competitive displacement assay as previously described in Neumeyer (Journal o...More data for this Ligand-Target Pair
Affinity DataEC50: 4.80nMpH: 7.4Assay Description:The EC50 and Imax for μ opioid receptors was determined using a [I35S]GTPγS binding assay. This assay measures the functional properties of a compo...More data for this Ligand-Target Pair