BDBM136287 US8853212, DDP-4 Inhibitor 3::US8853212, DDP-4 Inhibitor 4

SMILES N[C@H]1C[C@H](CS(=O)C1c1cc(F)cc(F)c1F)N1Cc2c[nH]nc2C1

InChI Key

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 136287   

TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM136287(US8853212, DDP-4 Inhibitor 3 | US8853212, DDP-4 I...)
Affinity DataIC50:  49nMpH: 7.5Assay Description:A continuous fluorometric assay is employed with the substrate Gly-Pro-AMC, which is cleaved by DPP-4 to release the fluorescent AMC leaving group. T...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM136287(US8853212, DDP-4 Inhibitor 3 | US8853212, DDP-4 I...)
Affinity DataIC50:  40nMpH: 7.5Assay Description:A continuous fluorometric assay is employed with the substrate Gly-Pro-AMC, which is cleaved by DPP-4 to release the fluorescent AMC leaving group. T...More data for this Ligand-Target Pair
In DepthDetails US Patent