BDBM138071 US8871934, 664
SMILES [#6]\[#6](-[#6])=[#6]/c1cc2c(-c3ccccc3C2([#8])C(F)(F)F)c(c1)-c1cnn(c1)-[#6](-[#6]-[#8])-[#6]-[#8]
InChI Key InChIKey=QLFQBMDXKHYFGU-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 138071
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 2, mitochondrial(Homo sapiens (Human))
Japan Tobacco
US Patent
Japan Tobacco
US Patent
Affinity DataIC50: 15nMpH: 8.0 T: 2°CAssay Description:The inhibitory action of PDHK activity was indirectly evaluated by performing a kinase reaction in the presence of a test compound and measuring the ...More data for this Ligand-Target Pair