BDBM20478 1-(2-bromophenyl)-3-{2-[(3-methylphenyl)amino]ethyl}urea::urea TRPV1 antagonist, 11

SMILES Cc1cccc(NCCNC(=O)Nc2ccccc2Br)c1

InChI Key InChIKey=ZHIILYBYAZTTPK-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 20478   

LigandPNGBDBM20478(1-(2-bromophenyl)-3-{2-[(3-methylphenyl)amino]ethy...)
Affinity DataEC50: >158nMpH: 7.2 T: 2°CAssay Description:One day before the assay was performed, human TRPV1 expressed in 1321N1 astrocytoma cells were plated onto 96-well assay plates and grown until 2.5 h...More data for this Ligand-Target Pair
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