BDBM264523 7-[3,5- bis(trifluoromethyl)phenyl]- 4-({2-(dimethylamino)-5-[4- fluoro-2-methoxy-5-(1- methylethyl)phenyl] pyrimidin-4-yl} methyl)-6-oxa-4- azaspiro[2.4]heptan-5-one::US9717714, 10
SMILES COc1cc(F)c(cc1-c1cnc(nc1CN1C(=O)OC(c2cc(cc(c2)C(F)(F)F)C(F)(F)F)C11CC1)N(C)C)C(C)C
InChI Key InChIKey=GVRLSMLSQQDGKB-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 264523
Affinity DataIC50: 345nMAssay Description:Transfer assays are performed in a 96-well v-bottom polypropylene plate. For the RTA using recombinant CETP (2% RTA), an assay cocktail is prepared w...More data for this Ligand-Target Pair