BDBM28683 2-({3-[(4-bromo-1H-indole-1-)sulfonyl]benzene}amido)-5-methylbenzoic acid::Anthranilic acid deriv., 21

SMILES Cc1ccc(NC(=O)c2cccc(c2)S(=O)(=O)n2ccc3c(Br)cccc23)c(c1)C(O)=O

InChI Key InChIKey=IJPGVCVMSQNPSN-UHFFFAOYSA-N

Data  9 IC50  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 9 hits for monomerid = 28683   

LigandPNGBDBM28683(2-({3-[(4-bromo-1H-indole-1-)sulfonyl]benzene}amid...)
Affinity DataIC50:  10nM EC50:  13nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28683(2-({3-[(4-bromo-1H-indole-1-)sulfonyl]benzene}amid...)
Affinity DataIC50:  1.26E+3nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28683(2-({3-[(4-bromo-1H-indole-1-)sulfonyl]benzene}amid...)
Affinity DataIC50:  1.26E+3nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28683(2-({3-[(4-bromo-1H-indole-1-)sulfonyl]benzene}amid...)
Affinity DataIC50:  1.26E+3nMAssay Description:Agonist activity at PPARalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28683(2-({3-[(4-bromo-1H-indole-1-)sulfonyl]benzene}amid...)
Affinity DataIC50:  1.26E+3nMAssay Description:Agonist activity at PPARgammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28683(2-({3-[(4-bromo-1H-indole-1-)sulfonyl]benzene}amid...)
Affinity DataIC50:  1.26E+3nMAssay Description:Agonist activity at PPARgammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28683(2-({3-[(4-bromo-1H-indole-1-)sulfonyl]benzene}amid...)
Affinity DataIC50:  1.26E+3nMAssay Description:Agonist activity at PPARalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28683(2-({3-[(4-bromo-1H-indole-1-)sulfonyl]benzene}amid...)
Affinity DataIC50:  10nMAssay Description:Agonist activity at PPARdeltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28683(2-({3-[(4-bromo-1H-indole-1-)sulfonyl]benzene}amid...)
Affinity DataIC50:  10nMAssay Description:Agonist activity at PPARdeltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed