BDBM311803 7-Chloro-8-(7-chloro-1H-indazol-5-yl)-2-(trifluoromethyl)-[1,2,4]triazolo[1,5-a]pyridine::US10155769, Example 41

SMILES FC(F)(F)c1nc2c(c(Cl)ccn2n1)-c1cc(Cl)c2[nH]ncc2c1

InChI Key InChIKey=GYKVBSCJPHIEQL-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 311803   

TargetVoltage-dependent calcium channel gamma-2 subunit(Human)
Janssen Pharmaceutica

US Patent
LigandPNGBDBM311803(US10155769, Example 41 | 7-Chloro-8-(7-chloro-1H-i...)
Affinity DataIC50: 1nMAssay Description:An in vitro assay was used to determine the potency of test compounds as inhibitors of the glutamate response of the channel formed by GluA1o-γ8...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent