BDBM458133 US10752616, Code No. BHBA-005

SMILES Cc1ccc(C)c2oc(cc12)-c1nc(no1)-c1ccc(cc1N)C(O)=O

InChI Key InChIKey=VYNIAJAXQZQNPS-UHFFFAOYSA-N

Data  3 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 458133   

TargetRetinoic acid receptor beta(Homo sapiens (Human))
King''S College London

US Patent
LigandPNGBDBM458133(US10752616, Code No. BHBA-005)
Affinity DataEC50:  23nMAssay Description:Transcriptional transactivation assays were performed with gal4 fusion receptor constructs, created using each of the RAR ligand binding domains of e...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
King''S College London

US Patent
LigandPNGBDBM458133(US10752616, Code No. BHBA-005)
Affinity DataEC50:  55nMAssay Description:Transcriptional transactivation assays were performed with gal4 fusion receptor constructs, created using each of the RAR ligand binding domains of e...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
King''S College London

US Patent
LigandPNGBDBM458133(US10752616, Code No. BHBA-005)
Affinity DataEC50:  130nMAssay Description:Transcriptional transactivation assays were performed with gal4 fusion receptor constructs, created using each of the RAR ligand binding domains of e...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent