BDBM494129 N-[6-[4-(2- amino-2-oxo- ethyl)piperazin- 1-yl]-1-oxo-2- tetrahydropyran- 4-yl-isoindolin- 5- yl]pyrazolo[1,5- a]pyrimidine-3- carboxamide::US10988478, Example 177

SMILES NC(=O)CN1CCN(CC1)c1cc2C(=O)N(Cc2cc1NC(=O)c1cnn2cccnc12)C1CCOCC1

InChI Key InChIKey=GVHMANCGTYWJBE-UHFFFAOYSA-N

Data  1 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 494129   

TargetInterleukin-1 receptor-associated kinase 4(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM494129(N-[6-[4-(2- amino-2-oxo- ethyl)piperazin- 1-yl]-1-...)
Affinity DataKi:  2nMAssay Description:Kinase activities were assayed using the Transcreener-Fluorecescence polarization platform (BelBrook Labs, Madison, Wis., USA) that measures amounts ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent