BDBM50015198 CHEMBL3262428

SMILES CN(CCCCN1CCN(CC1)c1ccccc1)c1cccc(O)c1

InChI Key InChIKey=ONEQFEKVBZHFKR-UHFFFAOYSA-N

Data  1 KI  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50015198   

Target5-hydroxytryptamine receptor 7(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50015198(CHEMBL3262428)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]5-HT from human 5-HT7 receptor expressed in HEK293 cells after 30 mins by microbeta counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50015198(CHEMBL3262428)
Affinity DataIC50: 540nMAssay Description:Antagonist activity at human 5-HT7 receptor expressed in CHO cells assessed as inhibition of 5-HT-stimulated cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed