BDBM50080334 (R)-1-{2-[1-(3-Methyl-thiophen-2-yl)-1-thiophen-2-yl-meth-(Z)-ylideneaminooxy]-ethyl}-piperidine-3-carboxylic acid; hydrochloride::CHEMBL543400
SMILES Cc1ccsc1\C(=N/OCCN1CCC[C@H](C1)C(O)=O)c1cccs1
InChI Key InChIKey=MKTBEDWVRUJECW-DZTQIWHNSA-N
Data 1 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 50080334
TargetSodium- and chloride-dependent GABA transporter 1(Rattus norvegicus)
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataKi: 74nMAssay Description:In vitro inhibition of [3H]GABA uptake at the Sodium- and chloride-dependent GABA transporter 1 (GAT-1) uptake site in rat brain synaptosomesMore data for this Ligand-Target Pair