BDBM50232047 CHEMBL4074253
SMILES CCCn1c(=O)n(CC)c2nc([nH]c2c1=O)-c1cnn(CC2CN(C(=O)C2)c2ccc(cc2)C(F)(F)F)c1
InChI Key InChIKey=VTWJQIYQJKMCSP-UHFFFAOYSA-N
Data 5 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 50232047
Affinity DataKi: 4nMAssay Description:Displacement of [3H]-MRS-1754 from human adenosine receptor A2b expressed in HEK293 cell membranes after 90 mins by liquid scintillation counting met...More data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Antagonist activity at human adenosine receptor A2b expressed in HEK293 cells assessed as inhibition of NECA-induced cAMP level preincubated for 15 m...More data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in HEK293 cells assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
Affinity DataKi: 460nMAssay Description:Displacement of [3H]-ZM-241385 from human adenosine receptor A2a expressed in HEK293 cell membranes after 90 mins by liquid scintillation counting me...More data for this Ligand-Target Pair
Affinity DataKi: 670nMAssay Description:Displacement of [3H]DPCPX from human adenosine receptor A1 expressed in HEK293 cell membranes after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair