BDBM50246776 3-(1,3-Dioxo-1,3-dihydro-2H-indolo[1',7':4,5,6]pyrrolo[3',4':2,3][1,4]diazepino[1,7-a]indol-2-yl)propyl N-Methylimidothiocarbamate::CHEMBL488271
SMILES CN=C(N)SCCCn1c(=O)c2c(n3c(cc4ccccc34)c3cccc4ccn2c34)c1=O
InChI Key InChIKey=MTYBEFAXRMHIIW-UHFFFAOYSA-N
Data 8 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 8 hits for monomerid = 50246776
Affinity DataIC50: 6.30E+3nMAssay Description:Inhibition of human INSRMore data for this Ligand-Target Pair
TargetNUAK family SNF1-like kinase 1(Homo sapiens (Human))
Institute Of General Genetics
Curated by ChEMBL
Institute Of General Genetics
Curated by ChEMBL
Affinity DataIC50: 9.70E+3nMAssay Description:Inhibition of human ARK5More data for this Ligand-Target Pair
Affinity DataIC50: 6.20E+3nMAssay Description:Inhibition of human CDK4/CycD1More data for this Ligand-Target Pair
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of human EPHB4More data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Institute Of General Genetics
Curated by ChEMBL
Institute Of General Genetics
Curated by ChEMBL
Affinity DataIC50: 7.40E+3nMAssay Description:Inhibition of human METMore data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor beta(Homo sapiens (Human))
Institute Of General Genetics
Curated by ChEMBL
Institute Of General Genetics
Curated by ChEMBL
Affinity DataIC50: 6.70E+3nMAssay Description:Inhibition of human PDGFRbetaMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Institute Of General Genetics
Curated by ChEMBL
Institute Of General Genetics
Curated by ChEMBL
Affinity DataIC50: 9.90E+3nMAssay Description:Inhibition of human EGFRMore data for this Ligand-Target Pair
Affinity DataIC50: 6.30E+3nMAssay Description:Inhibition of human CDK2/Cyc2More data for this Ligand-Target Pair