BDBM50254249 (5S)-5-[(4R)-4-{[(1-benzoylpiperidin-4-yl)carbonyl]amino}-3-oxo-3,4,5,10-tetrahydroazepino[3,4-b]indol-2(1H)-yl]-6-(benzylamino)-6-oxohexan-1-aminium trifluoroacetate::CHEMBL454202

SMILES NCCCC[C@H](N1Cc2[nH]c3ccccc3c2C[C@@H](NC(=O)C2CCN(CC2)C(=O)c2ccccc2)C1=O)C(=O)NCc1ccccc1

InChI Key InChIKey=QVYAOFKXMBYFNP-CWTKIQHKSA-N

Data  5 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50254249   

TargetSomatostatin receptor type 4(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50254249((5S)-5-[(4R)-4-{[(1-benzoylpiperidin-4-yl)carbonyl...)
Affinity DataIC50:  6.90nMAssay Description:Displacement of [125I]-[Leu8, DTrp22, Tyr25]-somatostatin-28 from human recombinant sst4 receptor expressed in chinese hamster CCL39 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50254249((5S)-5-[(4R)-4-{[(1-benzoylpiperidin-4-yl)carbonyl...)
Affinity DataIC50:  1.40nMAssay Description:Displacement of [125I]-[Leu8, DTrp22, Tyr25]-somatostatin-28 from human recombinant sst5 receptor expressed in chinese hamster CCL39 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50254249((5S)-5-[(4R)-4-{[(1-benzoylpiperidin-4-yl)carbonyl...)
Affinity DataIC50:  119nMAssay Description:Displacement of [125I]-[Leu8, DTrp22, Tyr25]-somatostatin-28 from human recombinant sst3 receptor expressed in chinese hamster CCL39 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50254249((5S)-5-[(4R)-4-{[(1-benzoylpiperidin-4-yl)carbonyl...)
Affinity DataIC50:  2.10nMAssay Description:Displacement of [125I]-[Leu8, DTrp22, Tyr25]-somatostatin-28 from human recombinant sst2 receptor expressed in chinese hamster CCL39 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50254249((5S)-5-[(4R)-4-{[(1-benzoylpiperidin-4-yl)carbonyl...)
Affinity DataIC50:  89nMAssay Description:Displacement of [125I]-[Leu8, DTrp22, Tyr25]-somatostatin-28 from human recombinant sst1 receptor expressed in chinese hamster CCL39 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed