BDBM50260199 CHEMBL4066038

SMILES COc1cc(OC)c(Cl)c(N2Cc3cnc(Nc4cc(F)cc(F)c4)nc3N(C3CCN(CC3)C(=O)\C=C\CN(C)C)C2=O)c1Cl

InChI Key InChIKey=UMIVIWIXPXKSIW-AATRIKPKSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50260199   

TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Guangzhou Institutes of Biomedicine and Health

Curated by ChEMBL
LigandPNGBDBM50260199(CHEMBL4066038)
Affinity DataIC50:  1.80nMAssay Description:Inhibition of human recombinant His-tagged FGFR1 cytoplasmic domain (308 to 731 residues) expressed in baculovirus using Tyr-4 peptide after 1 hr by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed