BDBM50266639 3-(2-(dimethylamino)ethyl)-2-methyl-N-(naphthalen-1-yl)-1H-indene-5-sulfonamide::CHEMBL475969

SMILES CN(C)CCC1=C(C)Cc2ccc(cc12)S(=O)(=O)Nc1cccc2ccccc12

InChI Key InChIKey=NCXJCTGPMJFTES-UHFFFAOYSA-N

Data  2 IC50  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50266639   

Target5-hydroxytryptamine receptor 6(Human)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50266639(3-(2-(dimethylamino)ethyl)-2-methyl-N-(naphthalen-...)
Affinity DataEC50:  14nMAssay Description:Agonist activity at human 5HT6 receptor expressed in HEK293F cells assessed as stimulation of cAMP level after 30 mins by HTRF assay Inhibition of ra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50266639(3-(2-(dimethylamino)ethyl)-2-methyl-N-(naphthalen-...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human 5HT1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2012
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50266639(3-(2-(dimethylamino)ethyl)-2-methyl-N-(naphthalen-...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human adrenergic alpha2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2012
Entry Details Article
PubMed