BDBM50339761 CHEMBL1689109::[4-Chloro-2-[4-(phenylsulfonyl)-1-piperazinylmethyl]phenoxy]-acetic acid
SMILES OC(=O)COc1ccc(Cl)cc1CN1CCN(CC1)S(=O)(=O)c1ccccc1
InChI Key InChIKey=VEDPQGGGGHKSLY-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50339761
Affinity DataIC50: 16nMAssay Description:Displacement of [3H]PGD2 from human CRTh2 receptor expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 201nMAssay Description:Antagonist activity against human CRTh2 receptor expressed in CHO cells assessed as inhibition of PGD2-mediated Ca2+ fluxMore data for this Ligand-Target Pair