BDBM50381771 CHEMBL2023457

SMILES COc1ccc2c(ccnc2c1)-c1cnn(c1)-c1ccccc1

InChI Key InChIKey=WSCLENBLVSFSQG-UHFFFAOYSA-N

Data  1 IC50  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50381771   

TargetMetabotropic glutamate receptor 4(Human)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50381771(CHEMBL2023457)
Affinity DataEC50:  220nMAssay Description:Positive allosteric modulation of human mGlu4 receptor expressed in BHK cells assessed as potentiation of glutamate-induced calcium mobilization by F...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50381771(CHEMBL2023457)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of human ERG by electrophysiology assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed