BDBM50469400 CHEMBL4278109

SMILES CCCc1nc2c(C)cccc2n1Cc1ccc2c(COc3ccccc3\C2=C(/C)c2noc(=O)[nH]2)c1

InChI Key InChIKey=KWALRLFFHWLMRU-ZXVVBBHZSA-N

Data  2 EC50

PDB links: 1 PDB ID matches this monomer.

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50469400   

TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50469400(CHEMBL4278109)
Affinity DataEC50:  3.30nMAssay Description:Agonist activity at PPARgamma in human MKN45 cells assessed as induction of cell aggregation incubated for 5 days by Hoechst 33342 staining based IN ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50469400(CHEMBL4278109)
Affinity DataEC50:  2.40nMAssay Description:Transactivation of GAL4-fused human PPARgamma transfected in HEK293BENA cells after 24 hrs by steady glo-luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB