BDBM50576716 CHEMBL4870494
SMILES CC1COc2c(N3CCN(C)CC3)c(F)cc3c2n1cc(C(=O)N(C)CCCN1c2ccccc2CCc2ccccc12)c3=O
InChI Key InChIKey=WARTVLAEBFUNAM-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50576716
TargetBromodomain-containing protein 4(Homo sapiens (Human))
The University Of Hong Kong
Curated by ChEMBL
The University Of Hong Kong
Curated by ChEMBL
Affinity DataIC50: 4.10E+4nMAssay Description:Displacement of SGRG-K(Ac)-GG-K(Ac)-GLG-K(Ac)-GGA-K(Ac)-RHRKVGG-K(Biotin) from Europium chelated human BRD4 bromodomain 2 (342 to 460 residues) measu...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
The University Of Hong Kong
Curated by ChEMBL
The University Of Hong Kong
Curated by ChEMBL
Affinity DataIC50: 2.27E+5nMAssay Description:Displacement of SGRG-K(Ac)-GG-K(Ac)-GLG-K(Ac)-GGA-K(Ac)-RHRKVGG-K(Biotin) from Europium chelated human BRD4 bromodomain 1 (49 to 170 residues) measur...More data for this Ligand-Target Pair