BDBM587732 2-[({5-[(2-methylbiphenyl-3-yl)amino]pyrido[3,4-b]pyrazin-2-yl}methyl)amino]ethanol::US11535615, Example 14

SMILES Cc1c(Nc2nccc3nc(CNCCO)cnc23)cccc1-c1ccccc1

InChI Key InChIKey=PISXMONKQHOZNA-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 587732   

TargetProgrammed cell death 1 ligand 1 [19-238]/protein 1 [25-167](Homo sapiens (Human))
Incyte

US Patent
LigandPNGBDBM587732(2-[({5-[(2-methylbiphenyl-3-yl)amino]pyrido[3,4-b]...)
Affinity DataIC50: <10nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails US Patent