BDBM283118 (R)-(6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-benzo[f][1,2,4]triazolo[4,3-a][1,4]diazepin-4-yl)methyl dimethylsulfamate ::US9884874, Compound 9
SMILES COc1ccc-2c(c1)C(=N[C@@H](COS(=O)(=O)N(C)C)c1nnc(C)n-21)c1ccc(Cl)cc1
InChI Key InChIKey=NEXIHPRJFHEPMD-SFHVURJKSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 283118
Affinity DataIC50: 280nMAssay Description:Bromodomain binding assays were carried out in Reaction Biology (PA, USA) to test the degrees of the inventive compounds in inhibiting the human BRD4...More data for this Ligand-Target Pair