BDBM28686 2-({3-[(5-chloro-1H-indole-1-)sulfonyl]benzene}amido)-5-methylbenzoic acid::Anthranilic acid deriv., 24

SMILES Cc1ccc(NC(=O)c2cccc(c2)S(=O)(=O)n2ccc3cc(Cl)ccc23)c(c1)C(O)=O

InChI Key InChIKey=LQDCBONSFOEGGS-UHFFFAOYSA-N

Data  9 IC50  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 9 hits for monomerid = 28686   

LigandPNGBDBM28686(2-({3-[(5-chloro-1H-indole-1-)sulfonyl]benzene}ami...)
Affinity DataIC50:  20nM EC50:  50nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28686(2-({3-[(5-chloro-1H-indole-1-)sulfonyl]benzene}ami...)
Affinity DataIC50:  2.00E+3nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28686(2-({3-[(5-chloro-1H-indole-1-)sulfonyl]benzene}ami...)
Affinity DataIC50:  1.59E+3nMAssay Description:Competition-binding curves for test compounds were determined with expressed human PPAR LBD. Plots of inhibitor concentration versus cpm of radioliga...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28686(2-({3-[(5-chloro-1H-indole-1-)sulfonyl]benzene}ami...)
Affinity DataIC50:  2.00E+3nMAssay Description:Agonist activity at PPARalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28686(2-({3-[(5-chloro-1H-indole-1-)sulfonyl]benzene}ami...)
Affinity DataIC50:  1.58E+3nMAssay Description:Agonist activity at PPARgammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28686(2-({3-[(5-chloro-1H-indole-1-)sulfonyl]benzene}ami...)
Affinity DataIC50:  2.00E+3nMAssay Description:Agonist activity at PPARalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28686(2-({3-[(5-chloro-1H-indole-1-)sulfonyl]benzene}ami...)
Affinity DataIC50:  20nMAssay Description:Agonist activity at PPARdeltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28686(2-({3-[(5-chloro-1H-indole-1-)sulfonyl]benzene}ami...)
Affinity DataIC50:  1.59E+3nMAssay Description:Agonist activity at PPARgammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM28686(2-({3-[(5-chloro-1H-indole-1-)sulfonyl]benzene}ami...)
Affinity DataIC50:  20nMAssay Description:Agonist activity at PPARdeltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed