BDBM311795 2-Methyl-8-(7-methyl-1H-indazol-5-yl)-7-(trifluoromethyl)-[1,2,4]triazolo[1,5-a]pyridine::US10155769, Example 33

SMILES Cc1nc2c(-c3cc(C)c4[nH]ncc4c3)c(ccn2n1)C(F)(F)F

InChI Key InChIKey=FELYLJINEBSAMA-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 311795   

TargetVoltage-dependent calcium channel gamma-2 subunit(Homo sapiens (Human))
Janssen Pharmaceutica

US Patent
LigandPNGBDBM311795(2-Methyl-8-(7-methyl-1H-indazol-5-yl)-7-(trifluoro...)
Affinity DataIC50:  12.6nMAssay Description:An in vitro assay was used to determine the potency of test compounds as inhibitors of the glutamate response of the channel formed by GluA1o-γ8...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent