BDBM336811 6-((((S)-1-amino-1-oxopropan- 2-yl)amino)methyl)-2-(4-(4- trifluoromethyl)phenoxy)cyclohex- 1-en-1-yl)pyrimidine- 4-carboxamide::US9745287, Compound 57
SMILES C[C@H](NCc1cc(nc(n1)C1=CCC(CC1)Oc1ccc(cc1)C(F)(F)F)C(N)=O)C(N)=O
InChI Key InChIKey=UDOHHODQWOMOFC-HKALDPMFSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 336811
Affinity DataKi: 175nMAssay Description:Cells Manual Electrophysiology: The hNav1.7 expressing HEK-293 cells are plated on 35 mm culture dishes pre-coated with poly-D-lysine in standard DME...More data for this Ligand-Target Pair
Affinity DataIC50: 557nMAssay Description:Assay Buffer: The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL...More data for this Ligand-Target Pair