BDBM344434 (S or R)-ethyl 3-((S)-4-((3-chloro- 1-ethyl-1H-pyrazol-4- yl)sulfonyl)-6-((((1,1,1-trifluoro- 2-methylpropan-2- yl)oxy)carbonyl)amino)-3,4- dihydro-2H-benzo[b][1,4]oxazin- 2-yl)-2-methylpropanoate::US9783511, 3E
SMILES CCOC(=O)[C@H](C)C[C@H]1CN(c2cc(NC(=O)OC(C)(C)C(F)(F)F)ccc2O1)S(=O)(=O)c1cn(CC)nc1Cl
InChI Key InChIKey=KQRAQWGQZXKLOI-ZBFHGGJFSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 344434
Affinity DataIC50: 6nMAssay Description:To identify novel antagonists of RORgammaT, an assay was developed which employs the interaction of RORgammaT with its co-activator peptide SRC1_2. T...More data for this Ligand-Target Pair