BDBM355794 3-(1,3-Benzothiazol-6-yl)-N-cyclopropyl-3H-imidazo[4,5-b]pyridine-2-carboxamide::US9815832, 71

SMILES O=C(NC1CC1)c1nc2cccnc2n1-c1ccc2ncsc2c1

InChI Key InChIKey=RIMSLYGHGHUFCL-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 355794   

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D(Homo sapiens (Human))
Pfizer

US Patent
LigandPNGBDBM355794(3-(1,3-Benzothiazol-6-yl)-N-cyclopropyl-3H-imidazo...)
Affinity DataIC50:  6.34E+3nMAssay Description:The PDE4B and 4D assays use scintillation proximity assay (SPA) technology to measure the inhibition of human recombinant PDE4B and PDE4D enzyme acti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Pfizer

US Patent
LigandPNGBDBM355794(3-(1,3-Benzothiazol-6-yl)-N-cyclopropyl-3H-imidazo...)
Affinity DataIC50:  155nMAssay Description:The PDE4B and 4D assays use scintillation proximity assay (SPA) technology to measure the inhibition of human recombinant PDE4B and PDE4D enzyme acti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent