BDBM372312 8-chloro-N-cyclobutyl- 7,9-dimethyl- pyrido[3',2':4,5]furo[3,2-d] pyrimidin-4-amine hydrochloride::US10239887, Cpd. No. 49

SMILES Cc1nc2oc3c(NC4CCC4)ncnc3c2c(C)c1Cl

InChI Key InChIKey=CURBYQKFAPXXTN-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 372312   

TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Vanderbilt University

US Patent
LigandPNGBDBM372312(8-chloro-N-cyclobutyl- 7,9-dimethyl- pyrido[3',2':...)
Affinity DataEC50:  695nMAssay Description:For high throughput measurement of agonist-evoked increases in intracellular calcium, CHO-K1 cells stably expressing muscarinic receptors were plated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent