BDBM50009105 CHEMBL3238305
SMILES CC#C[C@H]1CN(CCN1c1ccc(nc1)C(C)(O)C(F)(F)F)S(=O)(=O)c1ccc(N)nc1
InChI Key InChIKey=RXLXBIHPMQBGOC-FUKCDUGKSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50009105
Affinity DataEC50: 1.45E+3nMAssay Description:Inhibition of GKRP-GK interaction in mouse hepatocytes assessed as induction of GK translocation from nucleus to cytoplasm incubated for 20 mins prio...More data for this Ligand-Target Pair
Affinity DataIC50: 69nMAssay Description:Inhibition of biotin-tagged human GKRP/fluorescein-tagged GK interaction preincubated for 20 mins prior to GK addition measured after 2 to 4 hrs by A...More data for this Ligand-Target Pair