BDBM50087016 8-Acenaphthen-1-yl-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one::CHEMBL281274::Ro65-6570
SMILES O=C1NCN(c2ccccc2)C11CCN(CC1)C1Cc2cccc3cccc1c23
InChI Key InChIKey=BBOAHBVXCYBKLC-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 10 hits for monomerid = 50087016
Affinity DataKi: 0.520nMAssay Description:Competitive binding affinity against transfected HEK293 cells expressing human Opioid receptor like 1More data for this Ligand-Target Pair
Affinity DataKi: 5.90nMAssay Description:Competitive binding displacement analyses was performed from permanently transfected HEK293 cells expressing human Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Competitive binding displacement analyses was performed from permanently transfected HEK293 cells expressing Opioid receptor kappa 1More data for this Ligand-Target Pair
Affinity DataKi: 250nMAssay Description:Competitive binding displacement analyses was performed from permanently transfected HEK293 cells expressing human Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataEC50: 2.50E+3nMAssay Description:Effective concentration of the required to stimulate binding of GTPgammaS to mu1 receptor was determined using scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataEC50: 40nMAssay Description:Effective concentration required to stimulate binding of GTPgammaS to ORL1 receptor was determined using scintillation proximity assayMore data for this Ligand-Target Pair