BDBM50091034 CHEMBL3582121
SMILES CC1(C)Nc2c3CCCc3c(cc2C(C)(C)C1=O)-c1cncc2nccn12
InChI Key InChIKey=DEYFWGXTPWNADC-IBGZPJMESA-O
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50091034
Affinity DataKi: 46nMAssay Description:Displacement of [3H]-dexamethasone from cytosolic fraction of human recombinant glucocorticoid receptor by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: >1.25E+3nMAssay Description:Displacement of [3H]-progesterone from cytosolic fraction of human recombinant progesterone-B receptor by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: >3.33E+3nMAssay Description:Displacement of [3H]-aldosterone from cytosolic fraction of human recombinant mineralocorticoid receptor by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 93nMAssay Description:Antagonist activity at human glucocorticoid receptor transfected in CHOK1 cells assessed as inhibition of dexamethasone-induced receptor transcriptio...More data for this Ligand-Target Pair