BDBM50201344 CHEMBL238529::N-(3,4-dimethoxyphenyl)-1-methyl-4-(pyridin-4-ylmethylamino)-1H-imidazole-5-carboxamide

SMILES COc1ccc(NC(=O)c2c(NCc3ccncc3)ncn2C)cc1OC

InChI Key InChIKey=NBLCRYNLAHMCIA-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50201344   

TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Chemical Diversity

Curated by ChEMBL
LigandPNGBDBM50201344(CHEMBL238529 | N-(3,4-dimethoxyphenyl)-1-methyl-4-...)
Affinity DataIC50:  350nMAssay Description:Inhibition of VEGFR2 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Chemical Diversity

Curated by ChEMBL
LigandPNGBDBM50201344(CHEMBL238529 | N-(3,4-dimethoxyphenyl)-1-methyl-4-...)
Affinity DataIC50:  210nMAssay Description:Inhibition of VEGFR1 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Chemical Diversity

Curated by ChEMBL
LigandPNGBDBM50201344(CHEMBL238529 | N-(3,4-dimethoxyphenyl)-1-methyl-4-...)
Affinity DataIC50:  57nMAssay Description:Inhibition of VEGFR2 by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed