BDBM50209162 2-(4-methyl-piperazin-1-yl)-N-(3-thiophen-3-yl-2,4-dihydro-indeno[1,2-c]pyrazol-5-yl)-acetamide::CHEMBL245768

SMILES CN1CCN(CC(=O)Nc2cccc-3c2Cc2c-3n[nH]c2-c2ccsc2)CC1

InChI Key InChIKey=DQXRNJOFIYWUBI-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50209162   

TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209162(2-(4-methyl-piperazin-1-yl)-N-(3-thiophen-3-yl-2,4...)
Affinity DataIC50:  920nMAssay Description:Inhibition of KDR by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209162(2-(4-methyl-piperazin-1-yl)-N-(3-thiophen-3-yl-2,4...)
Affinity DataIC50:  4.33E+3nMAssay Description:Inhibition of c-Kit by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209162(2-(4-methyl-piperazin-1-yl)-N-(3-thiophen-3-yl-2,4...)
Affinity DataIC50:  710nMAssay Description:Inhibition of Flt1 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed