BDBM50387477 CHEMBL2047477

SMILES CCn1c2cccc3cccc(c23)\c1=C\[CH+]\C=c1/n(CC)c2cccc3cccc1c23

InChI Key InChIKey=FSOMZNMBKNFLGB-YFJQDTPYSA-N

Data  5 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50387477   

TargetProtein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50387477(CHEMBL2047477)
Affinity DataIC50:  4.10E+3nMAssay Description:Inhibition of His-tagged PRMT1 expressed in Escherichia coli BL21(DE3) cells using [14C]-S-adenosyl-L-methionine and histone H4 peptide after 8 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein arginine N-methyltransferase 3 [N508S](Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50387477(CHEMBL2047477)
Affinity DataIC50:  8.30E+3nMAssay Description:Inhibition of His6X-tagged PRMT3 expressed in Escherichia coli BL21(DE3) cells using [14C]-S-adenosyl-L-methionine and histone H4 peptide after 8 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-arginine methyltransferase CARM1(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50387477(CHEMBL2047477)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of GST-tagged CARM1 expressed in escherichia coli BL21(DE3) cells using using [14C]-S-adenosyl-L-methionine and histone H3 peptide after 8...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein arginine N-methyltransferase 6(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50387477(CHEMBL2047477)
Affinity DataIC50:  1.26E+4nMAssay Description:Inhibition of His6X-tagged PRMT6 expressed in Escherichia coli BL21(DE3) cells using [14C]-S-adenosyl-L-methionine and histone H4 peptide after 8 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50387477(CHEMBL2047477)
Affinity DataIC50:  9.10E+3nMAssay Description:Inhibition of His6X-tagged PRMT5 expressed in Escherichia coli BL21(DE3) cells using [14C]-S-adenosyl-L-methionine and histone H4 peptide after 8 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed