BDBM50423462 CHEMBL251835

SMILES CN1C[C@@H](C[C@H]2[C@H]1Cc1c(Br)[nH]c3cccc2c13)C(=O)N1CCN(CC1)c1ccc2nonc2c1

InChI Key InChIKey=GZFMZJDVLOZLLL-OMXJDXKCSA-N

Data  10 Kd

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 10 hits for monomerid = 50423462   

TargetSomatostatin receptor type 1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50423462(CHEMBL251835)
Affinity DataKd:  1.20nMAssay Description:Binding affinity to human recombinant sst1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50423462(CHEMBL251835)
Affinity DataKd:  6.46E+3nMAssay Description:Binding affinity to human recombinant sst5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(RAT)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50423462(CHEMBL251835)
Affinity DataKd:  0.372nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(RAT)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50423462(CHEMBL251835)
Affinity DataKd:  6.46E+3nMAssay Description:Displacement of [125I][Tyr3]octreotide from sst2 receptor in rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50423462(CHEMBL251835)
Affinity DataKd:  126nMAssay Description:Binding affinity to human dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50423462(CHEMBL251835)
Affinity DataKd:  6.76E+3nMAssay Description:Binding affinity to human recombinant sst2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50423462(CHEMBL251835)
Affinity DataKd:  3.63E+3nMAssay Description:Binding affinity to human recombinant sst4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50423462(CHEMBL251835)
Affinity DataKd:  2.34E+3nMAssay Description:Binding affinity to human recombinant sst3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50423462(CHEMBL251835)
Affinity DataKd:  78nMAssay Description:Binding affinity to human dopamine D4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50423462(CHEMBL251835)
Affinity DataKd:  28nMAssay Description:Binding affinity to human 5HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed