BDBM50429885 CHEMBL2333378

SMILES FC(F)(F)C(=O)c1ccc(cc1)C(=O)N1CCOc2ccc(cc2C1)-c1cn[nH]c1

InChI Key InChIKey=HGTXSCABVKRXHD-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50429885   

TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Exelixis

Curated by ChEMBL

LigandBDBM50429885(CHEMBL2333378)Copy SMILESCopy InChI

Affinity DataIC50:  1.05E+3nMAssay Description:Inhibition of PI3Kalpha (unknown origin) using PIP2 as substrate after 2 hrs by luminescence assayMore data for this Ligand-Target Pair

Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
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