Report error Found 154 with Last Name = 'brian jones' and Initial = 'a'
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Neurogen
Curated by ChEMBL
Neurogen
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced receptor activation by FLIPR assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Neurogen
Curated by ChEMBL
Neurogen
Curated by ChEMBL
Affinity DataIC50: 0.400nMAssay Description:Antagonist activity against low pH(5.0-5.5)-activated rat VR1More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Neurogen
Curated by ChEMBL
Neurogen
Curated by ChEMBL
Affinity DataIC50: 0.800nMAssay Description:Antagonist activity against capsaicin-activated human VR1 by FLIPR assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Neurogen
Curated by ChEMBL
Neurogen
Curated by ChEMBL
Affinity DataIC50: 0.800nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced receptor activation by FLIPR assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Neurogen
Curated by ChEMBL
Neurogen
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Antagonist activity against low pH(5.0-5.5)-activated rat VR1More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Neurogen
Curated by ChEMBL
Neurogen
Curated by ChEMBL
Affinity DataIC50: 1.10nMAssay Description:Antagonist activity against capsaicin-activated human VR1 by FLIPR assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Neurogen
Curated by ChEMBL
Neurogen
Curated by ChEMBL
Affinity DataIC50: 1.30nMAssay Description:Antagonist activity at Sprague-Dawley rat dorsal root ganglion TRPV1 assessed as inhibition of pH (5.0 to 5.5)-induced receptor activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Neurogen
Curated by ChEMBL
Neurogen
Curated by ChEMBL
Affinity DataIC50: 1.40nMAssay Description:Antagonist activity against low pH(5.0-5.5)-activated rat VR1More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Neurogen
Curated by ChEMBL
Neurogen
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Antagonist activity against low pH(5.0-5.5)-activated rat VR1More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Neurogen
Curated by ChEMBL
Neurogen
Curated by ChEMBL
Affinity DataIC50: 2.20nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced receptor activation by FLIPR assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Neurogen
Curated by ChEMBL
Neurogen
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Antagonist activity against capsaicin-activated human VR1 by FLIPR assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Neurogen
Curated by ChEMBL
Neurogen
Curated by ChEMBL
Affinity DataIC50: 3.20nMAssay Description:Antagonist activity at Sprague-Dawley rat dorsal root ganglion TRPV1 assessed as inhibition of pH (5.0 to 5.5)-induced receptor activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Neurogen
Curated by ChEMBL
Neurogen
Curated by ChEMBL
Affinity DataIC50: 3.20nMAssay Description:Antagonist activity at Sprague-Dawley rat dorsal root ganglion TRPV1 assessed as inhibition of pH (5.0 to 5.5)-induced receptor activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Neurogen
Curated by ChEMBL
Neurogen
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Antagonist activity against low pH(5.0-5.5)-activated rat VR1More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Neurogen
Curated by ChEMBL
Neurogen
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Antagonist activity against low pH(5.0-5.5)-activated rat VR1More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Neurogen
Curated by ChEMBL
Neurogen
Curated by ChEMBL
Affinity DataIC50: 4.40nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced receptor activation by FLIPR assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Neurogen
Curated by ChEMBL
Neurogen
Curated by ChEMBL
Affinity DataIC50: 4.60nMAssay Description:Antagonist activity at Sprague-Dawley rat dorsal root ganglion TRPV1 assessed as inhibition of pH (5.0 to 5.5)-induced receptor activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Neurogen
Curated by ChEMBL
Neurogen
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Antagonist activity against low pH(5.0-5.5)-activated rat VR1More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Neurogen
Curated by ChEMBL
Neurogen
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Antagonist activity against capsaicin-activated human VR1 by FLIPR assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Neurogen
Curated by ChEMBL
Neurogen
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Antagonist activity against low pH(5.0-5.5)-activated rat VR1More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Neurogen
Curated by ChEMBL
Neurogen
Curated by ChEMBL
Affinity DataIC50: 5.5nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced receptor activation by FLIPR assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Neurogen
Curated by ChEMBL
Neurogen
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Antagonist activity against capsaicin-activated human VR1 by FLIPR assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Neurogen
Curated by ChEMBL
Neurogen
Curated by ChEMBL
Affinity DataIC50: 6.30nMAssay Description:Antagonist activity at Sprague-Dawley rat dorsal root ganglion TRPV1 assessed as inhibition of pH (5.0 to 5.5)-induced receptor activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Neurogen
Curated by ChEMBL
Neurogen
Curated by ChEMBL
Affinity DataIC50: 7.10nMAssay Description:Antagonist activity at Sprague-Dawley rat dorsal root ganglion TRPV1 assessed as inhibition of pH (5.0 to 5.5)-induced receptor activationMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Neurogen
Curated by ChEMBL
Neurogen
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Antagonist activity against capsaicin-activated human VR1 by FLIPR assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Neurogen
Curated by ChEMBL
Neurogen
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Antagonist activity against low pH(5.0-5.5)-activated rat VR1More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Neurogen
Curated by ChEMBL
Neurogen
Curated by ChEMBL
Affinity DataIC50: 8.40nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced receptor activation by FLIPR assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Neurogen
Curated by ChEMBL
Neurogen
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Antagonist activity against low pH(5.0-5.5)-activated rat VR1More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Neurogen
Curated by ChEMBL
Neurogen
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Antagonist activity against low pH(5.0-5.5)-activated rat VR1More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Neurogen
Curated by ChEMBL
Neurogen
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Antagonist activity against capsaicin-activated human VR1 by FLIPR assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Neurogen
Curated by ChEMBL
Neurogen
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Antagonist activity against capsaicin-activated human VR1 by FLIPR assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Neurogen
Curated by ChEMBL
Neurogen
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Antagonist activity against low pH(5.0-5.5)-activated rat VR1More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Neurogen
Curated by ChEMBL
Neurogen
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced receptor activation by FLIPR assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Neurogen
Curated by ChEMBL
Neurogen
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Antagonist activity against low pH(5.0-5.5)-activated rat VR1More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Neurogen
Curated by ChEMBL
Neurogen
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced receptor activation by FLIPR assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Neurogen
Curated by ChEMBL
Neurogen
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Antagonist activity against capsaicin-activated human VR1 by FLIPR assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Neurogen
Curated by ChEMBL
Neurogen
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced receptor activation by FLIPR assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Neurogen
Curated by ChEMBL
Neurogen
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Antagonist activity against capsaicin-activated human VR1 by FLIPR assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Neurogen
Curated by ChEMBL
Neurogen
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Antagonist activity against low pH(5.0-5.5)-activated rat VR1More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Neurogen
Curated by ChEMBL
Neurogen
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Antagonist activity against capsaicin-activated human VR1 by FLIPR assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Neurogen
Curated by ChEMBL
Neurogen
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced receptor activation by FLIPR assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Neurogen
Curated by ChEMBL
Neurogen
Curated by ChEMBL
Affinity DataIC50: 26nMAssay Description:Antagonist activity against low pH(5.0-5.5)-activated rat VR1More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Neurogen
Curated by ChEMBL
Neurogen
Curated by ChEMBL
Affinity DataIC50: 27nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced receptor activation by FLIPR assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Neurogen
Curated by ChEMBL
Neurogen
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Antagonist activity against capsaicin-activated human VR1 by FLIPR assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Neurogen
Curated by ChEMBL
Neurogen
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced receptor activation by FLIPR assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Neurogen
Curated by ChEMBL
Neurogen
Curated by ChEMBL
Affinity DataIC50: 34nMAssay Description:Antagonist activity against low pH(5.0-5.5)-activated rat VR1More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Neurogen
Curated by ChEMBL
Neurogen
Curated by ChEMBL
Affinity DataIC50: 35nMAssay Description:Antagonist activity against low pH(5.0-5.5)-activated rat VR1More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Neurogen
Curated by ChEMBL
Neurogen
Curated by ChEMBL
Affinity DataIC50: 36nMAssay Description:Antagonist activity against low pH(5.0-5.5)-activated rat VR1More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Neurogen
Curated by ChEMBL
Neurogen
Curated by ChEMBL
Affinity DataIC50: 37nMAssay Description:Antagonist activity against low pH(5.0-5.5)-activated rat VR1More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Neurogen
Curated by ChEMBL
Neurogen
Curated by ChEMBL
Affinity DataIC50: 39nMAssay Description:Antagonist activity against capsaicin-activated human VR1 by FLIPR assayMore data for this Ligand-Target Pair