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Found 247 with Last Name = 'fulp' and Initial = 'a'
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

US Patent
LigandPNGBDBM192521(US9187480, 4-[8-(2-chlorophenyl)-9-(4-chlorophenyl...)
Affinity DataKi:  0.280nMAssay Description:Further characterization of select compounds was performed using radioligand displacement of [3H]1 and equilibrium dissociation constant (Ki) values ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

US Patent
LigandPNGBDBM50383388(CHEMBL2030738)
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H]SR141716 from human CB1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

US Patent
LigandPNGBDBM50399518(CHEMBL2180214)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

US Patent
LigandPNGBDBM192536(US9187480, N-{1-[8-(2-chlorophenyl)-9-(4-chlorophe...)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

US Patent
LigandPNGBDBM50399523(CHEMBL2180205)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

US Patent
LigandPNGBDBM192536(US9187480, N-{1-[8-(2-chlorophenyl)-9-(4-chlorophe...)
Affinity DataKi:  1.54nMAssay Description:Further characterization of select compounds was performed using radioligand displacement of [3H]1 and equilibrium dissociation constant (Ki) values ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

US Patent
LigandPNGBDBM50399534(CHEMBL2180215)
Affinity DataKi:  1.79nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

US Patent
LigandPNGBDBM192521(US9187480, 4-[8-(2-chlorophenyl)-9-(4-chlorophenyl...)
Affinity DataKi:  1.79nMAssay Description:Further characterization of select compounds was performed using radioligand displacement of [3H]1 and equilibrium dissociation constant (Ki) values ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

US Patent
LigandPNGBDBM50144618(CHEMBL3758534)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

US Patent
LigandPNGBDBM192534(US9187480, N-{1-[8-(2-chlorophenyl)-9-(4-chlorophe...)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

US Patent
LigandPNGBDBM192534(US9187480, N-{1-[8-(2-chlorophenyl)-9-(4-chlorophe...)
Affinity DataKi:  1.93nMAssay Description:Further characterization of select compounds was performed using radioligand displacement of [3H]1 and equilibrium dissociation constant (Ki) values ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

US Patent
LigandPNGBDBM192538(US9187480, N-{1-[8-(2-chlorophenyl)-9-(4-chlorophe...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

US Patent
LigandPNGBDBM192538(US9187480, N-{1-[8-(2-chlorophenyl)-9-(4-chlorophe...)
Affinity DataKi:  2.02nMAssay Description:Further characterization of select compounds was performed using radioligand displacement of [3H]1 and equilibrium dissociation constant (Ki) values ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

US Patent
LigandPNGBDBM192530(US9187480, N-{1-[8-(2-chlorophenyl)-9-(4-chlorophe...)
Affinity DataKi:  2.55nMAssay Description:Further characterization of select compounds was performed using radioligand displacement of [3H]1 and equilibrium dissociation constant (Ki) values ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

US Patent
LigandPNGBDBM50493599(CHEMBL2436755)
Affinity DataKi:  2.60nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

US Patent
LigandPNGBDBM192537(US9187480, N-{1-[8-(2-chlorophenyl)-9-(4-chlorophe...)
Affinity DataKi:  2.67nMAssay Description:Further characterization of select compounds was performed using radioligand displacement of [3H]1 and equilibrium dissociation constant (Ki) values ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

US Patent
LigandPNGBDBM192537(US9187480, N-{1-[8-(2-chlorophenyl)-9-(4-chlorophe...)
Affinity DataKi:  2.70nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

US Patent
LigandPNGBDBM50383402(CHEMBL2030754)
Affinity DataKi:  2.90nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

US Patent
LigandPNGBDBM192532(US9187480, N-{1-[8-(2-chlorophenyl)-9-(4-chlorophe...)
Affinity DataKi:  3.35nMAssay Description:Further characterization of select compounds was performed using radioligand displacement of [3H]1 and equilibrium dissociation constant (Ki) values ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

US Patent
LigandPNGBDBM192532(US9187480, N-{1-[8-(2-chlorophenyl)-9-(4-chlorophe...)
Affinity DataKi:  3.40nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

US Patent
LigandPNGBDBM50383388(CHEMBL2030738)
Affinity DataKi:  3.40nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

US Patent
LigandPNGBDBM50383388(CHEMBL2030738)
Affinity DataKi:  3.44nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

US Patent
LigandPNGBDBM192529(US9187480, ethyl N-{1-[8-(2-chlorophenyl)-9-(4-chl...)
Affinity DataKi:  3.57nMAssay Description:Further characterization of select compounds was performed using radioligand displacement of [3H]1 and equilibrium dissociation constant (Ki) values ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

US Patent
LigandPNGBDBM192529(US9187480, ethyl N-{1-[8-(2-chlorophenyl)-9-(4-chl...)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

US Patent
LigandPNGBDBM192535(US9187480, N-{1-[8-(2-chlorophenyl)-9-(4-chlorophe...)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

US Patent
LigandPNGBDBM192535(US9187480, N-{1-[8-(2-chlorophenyl)-9-(4-chlorophe...)
Affinity DataKi:  4.01nMAssay Description:Further characterization of select compounds was performed using radioligand displacement of [3H]1 and equilibrium dissociation constant (Ki) values ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

US Patent
LigandPNGBDBM192528(US9187480, N-tert-butyl-1-[8-(2-chlorophenyl)-9-(4...)
Affinity DataKi:  4.08nMAssay Description:Further characterization of select compounds was performed using radioligand displacement of [3H]1 and equilibrium dissociation constant (Ki) values ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

US Patent
LigandPNGBDBM192527(US9187480, N-{1-[8-(2-chlorophenyl)-9-(4-chlorophe...)
Affinity DataKi:  6nMAssay Description:Further characterization of select compounds was performed using radioligand displacement of [3H]1 and equilibrium dissociation constant (Ki) values ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

US Patent
LigandPNGBDBM192531(US9187480, 8-(2-chlorophenyl)-9-(4-chlorophenyl)-6...)
Affinity DataKi:  6.10nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

US Patent
LigandPNGBDBM192531(US9187480, 8-(2-chlorophenyl)-9-(4-chlorophenyl)-6...)
Affinity DataKi:  6.10nMAssay Description:Further characterization of select compounds was performed using radioligand displacement of [3H]1 and equilibrium dissociation constant (Ki) values ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

US Patent
LigandPNGBDBM50399531(CHEMBL2180218)
Affinity DataKi:  6.20nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

US Patent
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataKi:  6.20nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

US Patent
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataKi:  6.20nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

US Patent
LigandPNGBDBM192526(US9187480, N-{4-[8-(2-chlorophenyl)-9-(4-chlorophe...)
Affinity DataKi:  6.21nMAssay Description:Further characterization of select compounds was performed using radioligand displacement of [3H]1 and equilibrium dissociation constant (Ki) values ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

US Patent
LigandPNGBDBM50144619(CHEMBL3759785)
Affinity DataKi:  6.40nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

US Patent
LigandPNGBDBM50399533(CHEMBL2180216 | US9187480, tert-butyl N-{1-[8-(2-c...)
Affinity DataKi:  7.10nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

US Patent
LigandPNGBDBM50399533(CHEMBL2180216 | US9187480, tert-butyl N-{1-[8-(2-c...)
Affinity DataKi:  7.12nMAssay Description:Further characterization of select compounds was performed using radioligand displacement of [3H]1 and equilibrium dissociation constant (Ki) values ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

US Patent
LigandPNGBDBM50383386(CHEMBL2029362)
Affinity DataKi:  7.30nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

US Patent
LigandPNGBDBM50144614(CHEMBL3758884)
Affinity DataKi:  7.5nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

US Patent
LigandPNGBDBM50383399(CHEMBL2030751)
Affinity DataKi:  7.60nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

US Patent
LigandPNGBDBM50354809(CHEMBL1834021)
Affinity DataKi:  8nMAssay Description:Displacement of [3H]-SR141716A from human CB1 receptor expressed in CHO-K1 cells after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

US Patent
LigandPNGBDBM50144609(CHEMBL3759222)
Affinity DataKi:  8.80nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

US Patent
LigandPNGBDBM50383387(CHEMBL2030765)
Affinity DataKi:  9.20nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

US Patent
LigandPNGBDBM50144615(CHEMBL3759255)
Affinity DataKi:  9.20nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

US Patent
LigandPNGBDBM50144612(CHEMBL3759254)
Affinity DataKi:  9.60nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

US Patent
LigandPNGBDBM50399532(CHEMBL2180217)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

US Patent
LigandPNGBDBM50354809(CHEMBL1834021)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]-SR141716A from human CB1 receptor expressed in CHO-K1 cells after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

US Patent
LigandPNGBDBM192525(US9187480, 4-[8-(2-chlorophenyl)-9-(4-chlorophenyl...)
Affinity DataKi:  11nMAssay Description:Further characterization of select compounds was performed using radioligand displacement of [3H]1 and equilibrium dissociation constant (Ki) values ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

US Patent
LigandPNGBDBM50383413(CHEMBL2030933)
Affinity DataKi:  11.8nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Research Triangle Institute

US Patent
LigandPNGBDBM50140231(5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-4-meth...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]-SR141716A from human CB1 receptor expressed in CHO-K1 cells after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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