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Found 45 with Last Name = 'gianoncelli' and Initial = 'a'
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34046(iodinated benzimidazole, 9a)
Affinity DataKi:  19nM ΔG°:  -45.8kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34038(4,5,6,7-tetraiodobenzimidazole (TIBI), 1a)
Affinity DataKi:  23nM ΔG°:  -45.4kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34044(iodinated benzimidazole, 7a)
Affinity DataKi:  24nM ΔG°:  -45.2kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34051(iodinated benzimidazole, 14)
Affinity DataKi:  27nM ΔG°:  -44.9kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34052(iodinated benzimidazole, 15)
Affinity DataKi:  50nM ΔG°:  -43.3kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34054(iodinated benzimidazole, 17)
Affinity DataKi:  50nM ΔG°:  -43.3kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34053(iodinated benzimidazole, 16)
Affinity DataKi:  54nM ΔG°:  -43.2kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34048(iodinated benzimidazole, 11a)
Affinity DataKi:  70nM ΔG°:  -42.5kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34043(iodinated benzimidazole, 6a)
Affinity DataKi:  75nM ΔG°:  -42.3kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34050(iodinated benzimidazole, 13a)
Affinity DataKi:  90nM ΔG°:  -41.8kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34040(iodinated benzimidazole, 3a)
Affinity DataKi:  100nM ΔG°:  -41.6kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34047(iodinated benzimidazole, 10a)
Affinity DataKi:  120nM ΔG°:  -41.1kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34049(iodinated benzimidazole, 12a)
Affinity DataKi:  120nM ΔG°:  -41.1kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34056(iodinated benzimidazole, 23)
Affinity DataKi:  130nM ΔG°:  -40.9kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34055(iodinated benzimidazole, 21)
Affinity DataKi:  140nM ΔG°:  -40.7kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34039(iodinated benzimidazole, 2a)
Affinity DataKi:  160nM ΔG°:  -40.3kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34058(iodinated benzimidazole, 27)
Affinity DataKi:  160nM ΔG°:  -40.3kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34057(iodinated benzimidazole, 25)
Affinity DataKi:  180nM ΔG°:  -40.0kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34045(iodinated benzimidazole, 8a)
Affinity DataKi:  330nM ΔG°:  -38.5kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34041(iodinated benzimidazole, 4a)
Affinity DataKi:  460nM ΔG°:  -37.6kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34042(iodinated benzimidazole, 5a)
Affinity DataKi:  590nM ΔG°:  -37.0kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34059(brominated benzimidazole, 20)
Affinity DataKi:  1.34E+3nM ΔG°:  -34.9kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34060(brominated benzimidazole, 22)
Affinity DataKi:  1.45E+3nM ΔG°:  -34.7kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34062(brominated benzimidazole, 26)
Affinity DataKi:  1.51E+3nM ΔG°:  -34.6kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Rattus norvegicus (Rat))
University of Padova

LigandPNGBDBM34061(brominated benzimidazole, 24)
Affinity DataKi:  1.91E+3nM ΔG°:  -34.0kJ/molepH: 7.5 T: 2°CAssay Description:Inhibitory effect of test compound was assessed in reaction buffer containing purified CK2, synthetic peptide substrate, and [gamma-33P]ATP. Assays w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50094895(1,4-diamino-9,10-anthraquinone | 1,4-diamino-anthr...)
Affinity DataIC50:  330nMAssay Description:Inhibition of CK1deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50094893(1-Amino-4-hydroxy-anthraquinone | 1-hydroxy-4-amin...)
Affinity DataIC50:  660nMAssay Description:Inhibition of CK1deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50008516(IC261)
Affinity DataIC50:  1.24E+3nMAssay Description:Inhibition of CK1alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50008516(IC261)
Affinity DataIC50:  2.57E+3nMAssay Description:Inhibition of CK1deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHomeodomain-interacting protein kinase 2(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50094895(1,4-diamino-9,10-anthraquinone | 1,4-diamino-anthr...)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of HIPK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50094895(1,4-diamino-9,10-anthraquinone | 1,4-diamino-anthr...)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of DYRK1aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50094895(1,4-diamino-9,10-anthraquinone | 1,4-diamino-anthr...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of CK1alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50094893(1-Amino-4-hydroxy-anthraquinone | 1-hydroxy-4-amin...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of CK1alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Fgr(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50094895(1,4-diamino-9,10-anthraquinone | 1,4-diamino-anthr...)
Affinity DataIC50:  2.40E+4nMAssay Description:Inhibition of FgrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50094895(1,4-diamino-9,10-anthraquinone | 1,4-diamino-anthr...)
Affinity DataIC50:  2.47E+4nMAssay Description:Inhibition of PIM1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform gamma-1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50094893(1-Amino-4-hydroxy-anthraquinone | 1-hydroxy-4-amin...)
Affinity DataIC50:  2.62E+4nMAssay Description:Inhibition of CK1gamma1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform gamma-1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50094895(1,4-diamino-9,10-anthraquinone | 1,4-diamino-anthr...)
Affinity DataIC50:  3.40E+4nMAssay Description:Inhibition of CK1gamma1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50094895(1,4-diamino-9,10-anthraquinone | 1,4-diamino-anthr...)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of SykMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50094895(1,4-diamino-9,10-anthraquinone | 1,4-diamino-anthr...)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of LynMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase CSK(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50094895(1,4-diamino-9,10-anthraquinone | 1,4-diamino-anthr...)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of CSKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50240382(1,4-Dihydroxyanthrachinon | 1,4-dihydroxy-9,10-ant...)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of CK1alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform gamma-1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50240382(1,4-Dihydroxyanthrachinon | 1,4-dihydroxy-9,10-ant...)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of CK1gamma1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50240382(1,4-Dihydroxyanthrachinon | 1,4-dihydroxy-9,10-ant...)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of CK1deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50094895(1,4-diamino-9,10-anthraquinone | 1,4-diamino-anthr...)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of GST tagged ALKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform gamma-1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50008516(IC261)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of CK1gamma1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed