Compile Data Set for Download or QSAR
maximum 50k data
Found 137 with Last Name = 'ktorza' and Initial = 'a'
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM50030474(Avandamet | Avandaryl | Avandia | BRL-49653 | CHEB...)
Affinity DataKi:  8nM ΔG°:  -43.0kJ/molepH: 8.2 T: 2°CAssay Description:Binding assays were performed in 96-well plate format, using a classical filtration assay with a human full length PPARγ construct (GST-PPAR LBD...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM28681(5-[(4-{2-[methyl(pyridin-2-yl)amino]ethoxy}phenyl)...)
Affinity DataKi:  8nMAssay Description:Displacement of [3H]Rosiglitazone from human PPARgammaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM50234375((S)-2-ethoxy-3-(4-(2-(6-((methoxyimino)(phenyl)met...)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]Rosiglitazone from human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM28798((2S)-2-ethoxy-3-(4-{2-[4-(methanesulfonyloxy)pheny...)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]Rosiglitazone from human PPARgammaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM50294690((S)-2-ethoxy-3-(4-(2-(6-((methoxyimino)(phenyl)met...)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]rosiglitazone from human PPARgamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM50294688((S)-3-(4-(2-(6-((benzyloxyimino)(phenyl)methyl)-4,...)
Affinity DataKi:  18.4nMAssay Description:Displacement of [3H]rosiglitazone from human PPARgamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM50294692((S)-3-(4-(2-(6-((methoxyimino)(phenyl)methyl)-4,4-...)
Affinity DataKi:  33nMAssay Description:Displacement of [3H]rosiglitazone from human PPARgamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM50234377(2-ethoxy-3-(4-(2-(6-((methoxyimino)(phenyl)methyl)...)
Affinity DataKi:  48nMAssay Description:Displacement of [3H]Rosiglitazone from human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM50294691((S)-2-(2-benzoylphenylamino)-3-(4-(2-(6-((methoxyi...)
Affinity DataKi:  54nMAssay Description:Displacement of [3H]rosiglitazone from human PPARgamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM50294689((S)-3-(4-(2-(6-((allyloxyimino)(phenyl)methyl)-4,4...)
Affinity DataKi:  54.2nMAssay Description:Displacement of [3H]rosiglitazone from human PPARgamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM50234372((R)-2-ethoxy-3-(4-(2-(6-((methoxyimino)(phenyl)met...)
Affinity DataKi:  89nMAssay Description:Displacement of [3H]Rosiglitazone from human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM50294693((S)-3-(4-(2-(6-((cyclopropylmethoxyimino)(phenyl)m...)
Affinity DataKi:  254nMAssay Description:Displacement of [3H]rosiglitazone from human PPARgamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM233176(Sodium 8-hydroxy-8-(2-octyloxy-quinolin-3-yl)-oct-...)
Affinity DataKi:  378nM ΔG°:  -34.1kJ/molepH: 8.2 T: 2°CAssay Description:Binding assays were performed in 96-well plate format, using a classical filtration assay with a human full length PPARγ construct (GST-PPAR LBD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM233183(Sodium 8-hydroxy-8-(6-methoxy-2-pentyloxy-quinolin...)
Affinity DataKi:  583nM ΔG°:  -33.1kJ/molepH: 8.2 T: 2°CAssay Description:Binding assays were performed in 96-well plate format, using a classical filtration assay with a human full length PPARγ construct (GST-PPAR LBD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM50234373(CHEMBL253851 | ethyl 2-ethoxy-3-(4-(2-(6-((hydroxy...)
Affinity DataKi:  618nMAssay Description:Displacement of [3H]Rosiglitazone from human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM50172802(CHEMBL383607 | Sodium 8-hydroxy-8-(2-pentyloxy-qui...)
Affinity DataKi:  947nM ΔG°:  -32.0kJ/molepH: 8.2 T: 2°CAssay Description:Binding assays were performed in 96-well plate format, using a classical filtration assay with a human full length PPARγ construct (GST-PPAR LBD...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM233180(Sodium [5-hydroxy-5-(2-pentyloxy-quinolin-3-yl)-pe...)
Affinity DataKi:  1.93E+3nM ΔG°:  -30.3kJ/molepH: 8.2 T: 2°CAssay Description:Binding assays were performed in 96-well plate format, using a classical filtration assay with a human full length PPARγ construct (GST-PPAR LBD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM233181(Sodium [5-hydroxy-5-(2-methoxy-quinolin-3-yl)-pent...)
Affinity DataKi:  3.81E+3nM ΔG°:  -28.8kJ/molepH: 8.2 T: 2°CAssay Description:Binding assays were performed in 96-well plate format, using a classical filtration assay with a human full length PPARγ construct (GST-PPAR LBD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM50294695((S)-2-acetoxy-3-(4-(2-(6-((methoxyimino)(phenyl)me...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]rosiglitazone from human PPARgamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM50294694((S)-2-(2-ethoxy-2-oxoethylamino)-3-(4-(2-(6-((hydr...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]rosiglitazone from human PPARgamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM50234379(CHEMBL252995 | dimethyl 2-(4-(2-(6-benzoyl-4,4-dim...)
Affinity DataKi:  1.00E+4nMAssay Description:Displacement of [3H]Rosiglitazone from human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM50234378(CHEMBL399629 | ethyl 2-ethoxy-3-(4-(2-(6-((methoxy...)
Affinity DataKi:  1.00E+4nMAssay Description:Displacement of [3H]Rosiglitazone from human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM50234376(CHEMBL252996 | dimethyl 2-(4-(2-(6-((hydroxyimino)...)
Affinity DataKi:  1.00E+4nMAssay Description:Displacement of [3H]Rosiglitazone from human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM50234374((S)-ethyl 2-ethoxy-3-(4-(2-(6-((methoxyimino)(phen...)
Affinity DataKi:  1.00E+4nMAssay Description:Displacement of [3H]Rosiglitazone from human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM233184(Sodium 8-hydroxy-8-(2-pentyloxy-benzo[h]quinolin-3...)
Affinity DataKi: >1.00E+4nM ΔG°: >-26.5kJ/molepH: 8.2 T: 2°CAssay Description:Binding assays were performed in 96-well plate format, using a classical filtration assay with a human full length PPARγ construct (GST-PPAR LBD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM233182(8-Hydroxy-8-(2-pentyloxy-benzo[h]quinolin-3-yl)-oc...)
Affinity DataKi: >1.00E+4nM ΔG°: >-26.5kJ/molepH: 8.2 T: 2°CAssay Description:Binding assays were performed in 96-well plate format, using a classical filtration assay with a human full length PPARγ construct (GST-PPAR LBD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM233179(8-Hydroxy-8-(2-pentyloxy-quinolin-3-yl)-oct-5-ynoi...)
Affinity DataKi: >1.00E+4nM ΔG°: >-26.5kJ/molepH: 8.2 T: 2°CAssay Description:Binding assays were performed in 96-well plate format, using a classical filtration assay with a human full length PPARγ construct (GST-PPAR LBD...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM233178(Sodium 8-hydroxy-8-[2-(4,4,4-trifluoro-butoxy)-qui...)
Affinity DataKi: >1.00E+4nM ΔG°: >-26.5kJ/molepH: 8.2 T: 2°CAssay Description:Binding assays were performed in 96-well plate format, using a classical filtration assay with a human full length PPARγ construct (GST-PPAR LBD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM233177(Sodium 8-hydroxy-8-[2-(3-methoxy-propoxy)-quinolin...)
Affinity DataKi: >1.00E+4nM ΔG°: >-26.5kJ/molepH: 8.2 T: 2°CAssay Description:Binding assays were performed in 96-well plate format, using a classical filtration assay with a human full length PPARγ construct (GST-PPAR LBD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM233175(Sodium 8-hydroxy-8-(2-methoxy-quinolin-3-yl)-oct-5...)
Affinity DataKi: >1.00E+4nM ΔG°: >-26.5kJ/molepH: 8.2 T: 2°CAssay Description:Binding assays were performed in 96-well plate format, using a classical filtration assay with a human full length PPARγ construct (GST-PPAR LBD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM233174(8-Hydroxy-8-[2-(4,4,4-trifluoro-butoxy)-quinolin-3...)
Affinity DataKi: >1.00E+4nM ΔG°: >-26.5kJ/molepH: 8.2 T: 2°CAssay Description:Binding assays were performed in 96-well plate format, using a classical filtration assay with a human full length PPARγ construct (GST-PPAR LBD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM233173(8-Hydroxy-8-[2-(3-methoxy-propoxy)-quinolin-3-yl]-...)
Affinity DataKi: >1.00E+4nM ΔG°: >-26.5kJ/molepH: 8.2 T: 2°CAssay Description:Binding assays were performed in 96-well plate format, using a classical filtration assay with a human full length PPARγ construct (GST-PPAR LBD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM233172(8-Hydroxy-8-(2-octyloxy-quinolin-3-yl)-oct-5-ynoic...)
Affinity DataKi: >1.00E+4nM ΔG°: >-26.5kJ/molepH: 8.2 T: 2°CAssay Description:Binding assays were performed in 96-well plate format, using a classical filtration assay with a human full length PPARγ construct (GST-PPAR LBD...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit?? De Rennes 1

LigandPNGBDBM50172813(8-Hydroxy-8-(2-pentyloxy-quinolin-3-yl)-oct-5-ynoi...)
Affinity DataKi: >1.00E+4nM ΔG°: >-26.5kJ/molepH: 8.2 T: 2°CAssay Description:Binding assays were performed in 96-well plate format, using a classical filtration assay with a human full length PPARγ construct (GST-PPAR LBD...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM50234373(CHEMBL253851 | ethyl 2-ethoxy-3-(4-(2-(6-((hydroxy...)
Affinity DataEC50:  189nMAssay Description:Agonist activity at human PPARalpha by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM28798((2S)-2-ethoxy-3-(4-{2-[4-(methanesulfonyloxy)pheny...)
Affinity DataEC50:  414nMAssay Description:Agonist activity at human PPARalpha by GAL4 transactivation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM50234375((S)-2-ethoxy-3-(4-(2-(6-((methoxyimino)(phenyl)met...)
Affinity DataEC50:  7.90nMAssay Description:Agonist activity at human PPARalpha at 100 uM by GAL4 transactivation assay relative to WY 14,643More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM28681(5-[(4-{2-[methyl(pyridin-2-yl)amino]ethoxy}phenyl)...)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at human PPARalpha by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM50234377(2-ethoxy-3-(4-(2-(6-((methoxyimino)(phenyl)methyl)...)
Affinity DataEC50:  12nMAssay Description:Agonist activity at human PPARalpha by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM28798((2S)-2-ethoxy-3-(4-{2-[4-(methanesulfonyloxy)pheny...)
Affinity DataEC50:  37nMAssay Description:Agonist activity at human PPARalpha at 100 uM by GAL4 transactivation assay relative to WY 14,643More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM50234378(CHEMBL399629 | ethyl 2-ethoxy-3-(4-(2-(6-((methoxy...)
Affinity DataEC50:  19nMAssay Description:Agonist activity at human PPARalpha at 100 uM by GAL4 transactivation assay relative to WY 14,643More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM50234372((R)-2-ethoxy-3-(4-(2-(6-((methoxyimino)(phenyl)met...)
Affinity DataEC50:  65nMAssay Description:Agonist activity at human PPARalpha at 100 uM by GAL4 transactivation assay relative to WY 14,643More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM50234374((S)-ethyl 2-ethoxy-3-(4-(2-(6-((methoxyimino)(phen...)
Affinity DataEC50:  14nMAssay Description:Agonist activity at human PPARalpha at 100 uM by GAL4 transactivation assay relative to WY 14,643More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM50234374((S)-ethyl 2-ethoxy-3-(4-(2-(6-((methoxyimino)(phen...)
Affinity DataEC50:  29nMAssay Description:Agonist activity at human PPARalpha by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM50234372((R)-2-ethoxy-3-(4-(2-(6-((methoxyimino)(phenyl)met...)
Affinity DataEC50:  194nMAssay Description:Agonist activity at human PPARalpha by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM50234378(CHEMBL399629 | ethyl 2-ethoxy-3-(4-(2-(6-((methoxy...)
Affinity DataEC50:  30nMAssay Description:Agonist activity at human PPARalpha by GAL4 transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM28681(5-[(4-{2-[methyl(pyridin-2-yl)amino]ethoxy}phenyl)...)
Affinity DataEC50:  4nMAssay Description:Agonist activity at human PPARalpha at 100 uM by GAL4 transactivation assay relative to WY 14,643More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM50234376(CHEMBL252996 | dimethyl 2-(4-(2-(6-((hydroxyimino)...)
Affinity DataEC50:  195nMAssay Description:Agonist activity at human PPARalpha at 100 uM by GAL4 transactivation assay relative to WY 14,643More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM50234377(2-ethoxy-3-(4-(2-(6-((methoxyimino)(phenyl)methyl)...)
Affinity DataEC50:  11nMAssay Description:Agonist activity at human PPARalpha at 100 uM by GAL4 transactivation assay relative to WY 14,643More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Spot-Ea3857

Curated by ChEMBL
LigandPNGBDBM50234379(CHEMBL252995 | dimethyl 2-(4-(2-(6-benzoyl-4,4-dim...)
Affinity DataEC50:  152nMAssay Description:Agonist activity at human PPARalpha at 100 uM by GAL4 transactivation assay relative to WY 14,643More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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